This invention provides substituted cycloheptenes of the general formula I
##STR1##
in which
R.sup.1 represents OH, O-(C.sub.1 -C.sub.6)-alkyl, O-(C.sub.3
-C.sub.7)-cycloalkyl, O-aryl, C.sub.1 -C.sub.6 -alkyl-COO-, aryl-COO-,
R.sup.2 represents C.sub.1 -C.sub.6 -alkyl, (CH.sub.2).sub.(1-2) -aryl,
C.sub.2 -C.sub.6 -alkenyl-aryl and
R.sup.3 represents (CH.sub.2).sub.(0-1) -C.sub.5 -C.sub.7 -cycloalkyl,
(CH.sub.2).sub.(0-2) -aryl, heterocyclyl, C.sub.1 -C.sub.6
-alkyl-heterocyclyl
either as a racemate or in the form of the pure enantiomers, each as a base
or as a salt with a pharmaceutically acceptable acid, a process for their
preparation and their use as medicaments.
Этот вымысел обеспечивает замененные cycloheptenes вообще ## ## STR1 формулы iego в R.sup.1 представляет oh, O-(C.sub.1 - C.sub.6)-alkyl, O-(C.sub.3 - C.sub.7)-cycloalkyl, О-aril, C.sub.1 - C.sub.6 - alkyl-COO -, aryl-COO -, R.sup.2 представляет C.sub.1 - C.sub.6 - алкил, (CH.sub.2).sub.(1-2) - арил, C.sub.2 - C.sub.6 - алкенильн-aril и R.sup.3 представляют (CH.sub.2).sub.(0-1) - C.sub.5 - C.sub.7 - cycloalkyl, (CH.sub.2).sub.(0-2) - арил, heterocyclyl, C.sub.1 - C.sub.6 - alkil-heterocyclyl или как racemate или in the form of чисто энантиомеры, каждое как основание или как соль с фармацевтически приемлемо кислотой, процесс для их подготовки и их польза как medicaments.
