Substituted cyclic amine metalloprotease inhibitors

   
   

The invention provides compounds which are useful as inhibitors of metalloproteases, and which are effective in treating conditions characterized by excess activity of these enzymes. In particular, the present invention relates to a compound having a structure according to Formula (I). ##STR1## Also disclosed are compounds, pharmaceutical compositions and methods of treating diseases characterized by metalloprotease activity using these compounds or the pharmaceutical compositions containing them.

A invenção fornece os compostos que são úteis como inibidores dos metalloproteases, e que são eficazes nas circunstâncias de tratamento caracterizadas pela atividade adicional destes enzymes. No detalhe, a invenção atual relaciona-se a um composto que tem uma estrutura de acordo com a fórmula (i). ## do ## STR1 São divulgados também os compostos, as composições pharmaceutical e os métodos de tratar as doenças caracterizadas pela atividade do metalloprotease usando estes compostos ou as composições pharmaceutical que contêm os.

 
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< Insulin receptor-related receptor binding protein

< LFA-1 antagonist compounds

> Adenosine receptor ligands

> Phenyl-substituted indoles and indazoles

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