The present invention relates to a novel dibenzoxazepine derivative, its synthesis,
and its use as an v integrin receptor antagonist. More particularly, the
compound of the present invention is an antagonist of the integrin receptors v3
and v5 and therefor useful for inhibiting bone resorption, treating
and/or preventing osteoporosis, and inhibiting vascular restenosis, diabetic retinopathy,
macular degeneration, angiogenesis, artheroscietosis, inflammatory arthritis, cancer
and metastatic tumor growth.