The present invention discloses processes for preparing piperidine derivative
compounds of the formulae:
##STR1##
wherein
- n is 0 or 1;
- R1 is hydrogen or hydroxy;
- R2 is hydrogen;
- or, when n is 0, R1 and R2 taken together form
a second bond between the carbon atoms bearing R1 and R2,
provided that when n is 1, R1 and R2 are each hydrogen;
- R3 is —COOH or —COOR4;
- R4 is an alkyl or aryl moiety;
- A, B, and D are the substituents of their rings, each of which may be
different or the same, and are selected from the group consisting of hydrogen,
halogens, alkyl, hydroxy, alkoxy, and other substituents.
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