A process for preparing an optionally substituted
4-benzimidazol-2-ylmethylamino)benzamidine, the process comprising: (a)
condensing an optionally suitably substituted diaminobenzene with
2-[4-(1,2,4-oxadiazol-5-on-3-yl)phenylamino]acetic acid; (b)
hydrogenating the product obtained from step (a); and (c) optionally
carboxylating the amidino group of the product obtained from step (b).