An efficient synthesis for the preparation of
((1R,3S)-3-isopropyl-3-{[3-(trifluoromethyl)-7,8-dihydro-1,6-naphthyridin-
-6(5H)-yl]carbonyl}
cyclopentyl)[(3S,4S)-3-methoxytetrahydro-2H-pyran-4-yl]amine and its
succinate salt are provided. The succinate salt is crystalline and has
superior properties.