Compounds of formula (I) ##STR00001## wherein: X is CH or CH--R.sub.2;
R.sub.1 is C.sub.1-C.sub.6 linear or branched alkyl or C.sub.1-C.sub.6
linear or branched alkenyl; R.sub.2 is hydrogen, C.sub.1-C.sub.6 linear
or branched alkyl or C.sub.1-C.sub.6 linear or branched alkenyl,
C.sub.6-C.sub.14 aryl or C.sub.6-C.sub.14 aryl(C.sub.1-C.sub.6) linear or
branched alkyl or C.sub.6-C.sub.14 aryl(C.sub.1-C.sub.6) linear or
branched alkenyl, with the aryl group optionally substituted by one or
more substituents, either the same or different, selected from the group
consisting of halogen, hydroxy, C.sub.1-C.sub.6 alkoxy linear or branched
or C.sub.1-C.sub.6 alkenyloxy linear or branched, amino, optionally mono-
or disubstituted with C.sub.1-C.sub.6 linear or branched alkyl; R.sub.3
is NH.sub.2, or NHR.sub.4; R.sub.4 is C.sub.1-C.sub.6 alkyl or
C.sub.1-C.sub.6 hydroxyalkyl, C.sub.1-C.sub.3 alkoxyalkyl,
amino(C.sub.1-C.sub.6)alkyl, where the amino group is optionally
substituted with one or two C.sub.1-C.sub.3 linear or branched alkyl
groups, or with one or two C.sub.2-C.sub.3 alkenyl groups
C.sub.6-C.sub.14 aryl or C.sub.6-C.sub.14 aryl(C.sub.1-C.sub.6)alkyl,
with the aryl group optionally substituted by one or more substituents,
either the same or different, selected from the group consisting by
halogen, hydroxy, C.sub.1-C.sub.6 alkoxy linear or branched or
C.sub.1-C.sub.6 alkenyloxy linear or branched, amino, mono- or
di-substituted with C.sub.1-C.sub.6 alkyl linear or branched or
C.sub.1-C.sub.6 alkenyl linear or branched; and their pharmaceutically
acceptable salts. These compounds are antagonists of the adenosine
A.sub.2a receptor and useful as medicaments, in particular for the
treatment of Parkinson's disease.