Mono- and di-fluorinated benzothiepine compounds as inhibitors of apical sodium co-dependent bile acid transport (ASBT) and taurocholate uptake

   
   

Mono-flourinated and di-fluorinated benzothiepine apical sodium co-dependent bile acid transport (ASBT) inhibitors are disclosed together with methods of making the same, methods of using the same to treat hyperlipidemic conditions as well as pharmaceutical compositions containing the same compounds.

Gli inibitori co-dipendenti di trasporto dell'acido di bile del Mono-flourinated e sodio apical Di-fluorato di benzothiepine (ASBT) sono rilevati insieme ai metodi di fabbricazione dello stesso, metodi di usando lo stesso per trattare le circostanze iperlipidiche così come le composizioni farmaceutiche che contengono lo stesso residui.

 
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